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oro ~ i ~ praz6 - HH07 i" 000152 | } ~ Exygen, d Ri ARa%6-- 3407 \ TITLE HodofAoki fieDerm ofPectin cd (PFOA) Se \ AutHoR \ `EmilyDecker N\ DATEISSUED | \ January8, 2004 | \\ SPONSOR | `Haskell \Baboratoryafposor HiBealathxse o& Ens viroomental Sciences. Bo || ExypaReseach 305 | || hy EELS } BM008276Revi 2 a= `TOTALNUMBEROFPAGES || \\ 8 `Company Saniized.Doesnotcontaln TSCA CBI -- 000153 MANAGEMENTAPPROVAL I ou ERxesearch 7, EVixespFPlraeRsheiesdreotnyuch Date . sMhaaknKeeamdy fz Dus : Doron SponsorRepresentative Exygea Research | Pagezat20 000154 & I. B3 - `TABLE OF CONTENTS L SUMMARY eons . 3. CHEMICALSANDSUPPLIES ..cecossssssmmessmmeensnoeonon] F3.E3. EQUJANID SUPPPLIMEScEecvNerTcmresmesems-- essesseno on 8 3F 5. PREPARATION OFSTANDARDS An NDFORTIFICATIONSOLUTIONS corfc--e--cr--r--o--r----1 33..55.21..SFTOROTCIKFSIOCALTUITOINOSNOcLrUrTsIsOsNsS.s.s.sc smsmo eeoso eesr nor s os D 3.53.CALIBRATION STANDARDS ..T cerenrrnsmresmmeroore 10 4A2L.. PSLOAWDMIAPGRLAMEcPreRtOcrccCmeEosSrSoImeNnGemossommosio s er 10 10 43.SAMPLEPREPARATION recesses 45. Q4.U5A.N1.TLITCA/TMISO/NMc SSysteo mand Oe pezatineg eCoendeitsioenssvmmsoeemweoneorornroen111 44..5532..CTAULNIEBFRIALTEIOPNARPARMOECTEEDRSU.R.E.Sc __._.o .....____s ___.....m ..... co omms 1122 46. A4C5C4E.PTSAANMPCLEECRAINTAERLIYA.S.I.S. cee mommsmssesoonoseoees 1134 5. 44.87..TPIEMRERORREMQUAINRCEEDCFROIRTAENRAILAY.S.I.S...r momo en or ers1134. CALCULATIONS .o.eeesecemsmmmmsosmsesoes 15 6. SAFcmeETYcensoreens 13. Ey Research | Ps3ot20 000155 | LIST OFTABLES Table RecoveryofPFOAfrom FortificationsInMonkey SED......ceo.ecvnen 16 LISTOF FIGURES FFiigpuarne21..RPCaFplOirAbeawtaionihcuvrvCnegffoourLoP.oFfmOAaioCfontCroelrMoroMcoekskSepySurr ec Sempov leese1l7f FigurR e 3. RepresC entativeChioma stogamofa.10pp Sr tafonr PFdOAafa nCrodz Figor4e. ReiptrhesPeFntOaAtiavedChwriotmhaBtogLsam.ofoCfonStCrBoFlMOoAnr keySeerumFe ortifir edat10Ep0pt20 | EpaRemch Peet 000156 & | | ~ | | 1 SUMMARY `sTehrisumr,eport details amethodof analysisforperfluorooctancicacid (PFOA)in Toechericl fom of PFOA vs sein me `PQFuaOntAifiicsateixotnroafctPeFdOfAriosmacscoempmlisbheyd bpryoltieqiunipdrcehcirpoimtaattioongirnapshcyethoanmnitdaielsems, `spectrometry(LC/MS/MS)analyisusing selectedreactionmonitoring (SRM). sem. `Thelowerlimitofquantitation (LLOQ)forthismethodis10ppbforPOAin Quantificationis performed. singextractedcalibrationstandardscontainingan s"aThniismaethdovdiwiaosndfeovePloRpOeNdusingmonnkyecyasenrum.1T,h1e0ondvoperyceent rrecove]ry& 6.9%(Table T). A1.toRperpesrcenstcattaitvievceaclhbrroimoantocgarrvaemsfofrorPFPOFAOAi.mionnmkoetykseeyrusmerisumhaotwe.sihnoFviegsure Figures 2to 4. . Brg Rescarch Passer 000157 L 2. sergo e---------------- EXPERIMENTALCOMPOUNDS BCumcodNewne := opm homa FF F Hc Core = ompum1265 | HHA ~~ b | Fo[4 F F FF i | | Exygea Research. PagoGorzn 000158 3. CHEMICALSANDSUPPLIES 31. CCw aenels e cage "Methanol(MOE) Acetonitrile(ACN) Comalil ErTll artoenalAIOi `AmmoniumAcetate HPLC HPLC Reagent EMSceocs BM Science: Sigma-Aldrich JT90932 AX0145-1 A-1330 32. STANDARDS a ad Sl (PFOA) Tae Fay Se Products. 2afTQ H TMTDeR e perfluoroctancicacid, NA 9635 DuPont. Resi ----- . Page7020 -- 000159. 33.CETQrUIaePMEswNT AeNDSuEpepeLIyES Sow Sohcritceitg es STpoat -- CDFiErrNepoicecsGOgAL 1002000) arson DreamFnaysy Sraintteontfyopanrteeit oir KNepueme ES SRoni Sne ew( ndiHLrn, 2mLclearHPLCvial kit (cat# 5181-3400) vAaivoH:iPFaotnis eeeyEs ikomei m ny beei frd petiri timorn 1Noe Irr como, woopicava gy .D 5 oHeWPFrLsIei CrvecialosFfrItm oNrA(tuSmihbeetee Hssac,PpknLiepdCCed sasu,oe teotsced sa.m)p.lcecrmeuqstiT mnpootibne,musceed,iy PPE oi Eof 54CFTlihetm ynareestehnrdacsnetmxsnpsarmosve htsitstsoe wgidewieon r ome 24.Scumone 2 mn wewien is peur by ping || Nyete:T0hp.e1t 5d8ofammmongr io umacetati eandodiissoelo viongcn iindc1 cLsod ,f,OehonntiStateye Wsatet, n | Sop rete | .i 000160 @ || || | ~9 pr 35.PREPARATIONOFSTANDARDSAND FORTIFICATIONSOLUTIONS Analyt1.iscCaearbsubtmraanaidnaodrndsSsrt1aenuvdsaedrdd1fs0sc--atTlhhieesenetpseutrtdphoeasrreedsss:psonospeorefptahreeddetiecctoonrtrwolimdoinnkseyy 2. `Lacanoabnloyorscainst.aortyoCnosnctoamsosSppoinkdeisn--gTthoetsheefoLrtLiOfiQcattidons1a0exLuLsuOalQlyoprdeapaerwedesdt. 3. M1iancdteoitnxetSropmliimnkeeosnankaelTyyhsteiesceaulorr.etciofvceartyi.onsLareaprebparceoodnbtryroslpsiapkiiknegtsaortoeotprrhepyaeld seafmfpelceosfstthksnaomwpnlecmonactenitxroatniosnnsa.lMyiactalarescpoivkeecsy.aresso 19 evaluatth `Thesolutevolumesofthesiadardsmayb viedbyth analystsslong sth mcopoammyrebcoetepprpiirorfpenpaoporahtsrdrioseoserndsra1eydows.fdsoadonlngu.tae5tNtoohsteoolPvarelensptoaratarhetaimtoaanidndtniadtiincoeondns.c)eAnclttroeartnniaoctneesbormncsecnsitearoaryt.rnioyns1s P3r.o5.p1.eSrtioncdikvsiodluuatlisotnock solionsof ~ 100 gl. ofPFOA and "C- . EPpxuFrtcOiihtgAyes)rbtaonycdwkeds1iiol2gluhtueiiCn1o0gn1o1u06a0tmCa~L113w0i5imtmhsgmlaeoLtlfDheaPafnnEoaoblleyot1arimceaaaslx1)s0it0a.1nsdtaorvpdboee(lsc.uosomridreooencefst1deidpfencoassr.3 romthedatof preparation. 23.51.P2sr0.eF0pooarrteislfL.iocftafoitttniioaohfneiSvncooalPliuFioutnOimoAetsnsrtsoaeilndtaailrkodn.odfes1c0r0ibpediLn 3f.o5r.1PtFoOA1b00ymLilwting bod`PimrleLupwtaiirnsgh 1aaf0comerttLifiioccfattfihnoenvPstoCa-lnPduFamrOdeAostflfrulaii1sock0n.pgd/esmclr,ifbeodrfn"3C5P.F1O10A1b0y9 P0de.rs0oc0pr5eipbge/dimfLno.c3oi.f5f2iP.cCa2-i2oPdnFsO0a.A5nbmtyaLdiolofufttihneLg "O1pC0-0pPmF.lOAoffsootrlhuPerFiPOoFnAd.OecAsosenssoiinnoidnsogs @ P3r5o2p1s0f1o0c0lfmiLcawiiotnhsaacnctdoendiloefn0.31vpo/lumm.etfcfPkFOAcontsining e. dPeG 3isz5cp2ro ai1eb1e0m dif1no0a 30nm.c5Lt2iCwoiRnnthsdOst0aN.tn5dbmarrLdcodofifntii0nen0ag1vLopglO/ummmll.etosfsfoofrltuaPotsFiPoOFnAOdceAossncnbliendogin 005pg/mL.ofPC PFOAby diluting 0.1mL.ofthe FRO sonics orp omc Passer 000161 | | ~D @ { i | | d3e5s2crbi1b0edi1n003.a5..2 wi4t0h4a0c.t5omniLtdolfethine a"voCl-uPmFeOAsollusthio.n describedin bSotetpoleeasat)lisloftno2raiiCfcra0iwo6insctfhaontrdiamaredmsiatoxliutmnieuocnmespsiesnrraiyrotedofomifgae1kraytenoeaiwfsnrto1am2n5td-hamerLtdLotsDsnPogEf hestock sohuion. Ti3hd.e5en3tc.iacCaallllirtbocraottnihoesntaSsnatdmaapnrlddesasar.drs pTrhoecefsosrtitfhicraotiuognhtofhetxhet.rasctuinondparyocepdeupree,; `exactionsdoneaccording thefolowing ble: "ConMicxeOdF RoSroliuctaitoinon VFoorltmeeat(ilo)n VCaonmmosli `Sample(mL) EGaumro Calibentic Sunda! Ao0o-- 1 -- 050 --oT0-- 11r 02 --0 0l0011_ 210 a ooil o2m100 4. METHOD T4dheLsecrPiBrpotoiwowndDoifuaegoarcnahmasoepf.themetiodis given below,followedby | a dotaled Measure 0.1mL.soyfMss ameplp etF(luoshwiinDgioadign isrdpgaosmnaeblemiceopipete) Piapeii ncine LOM iaussi 42.SunProcesses Nosstibmepallelporwoecdetsoincoimspnleeetdlyedtfhoarws,ewriumdseam,plesr.ooHmotweems,pefvrzae,n Santisamsples EomResees Pugs 0ar20 000162 | & ~ & | ||1 43.SunPrzmancron s`tsoamrpeldexsemfiugsetcbaetetdhsohroouuglhdlaylsmoibxeedablelfoowreedtbeoienqguislaimbrpalteedtfoarroexotmrtacetmipone.rate. All 5a.cEp aoTcchobrar etcnhocfopsy naempepl(egesieexthiraohcstdedl(Ntybpbiscaxlw lym3d0torixnledscsop)uriansl t(ionsctludeaHtlreast CNai seciom`paica ayettrooe pFooal 1e ivetdy 3 rtoooonm Pr 1. Mesos0 mk.of \ le to 2a.rentcmt oct 2 3 (wcC v hiotdhmcaniaos lnyrto eawsxneeafdlesdes,i tncliosncelvoiedi,hae nnndvaoarmte,x ~1S02sedaconrdos). 0005 er 4. AnalyzesamplesusingelectrosprayLC/MS/MS. 45. QUANTITATION 45.1. LC/MS/MSSystemandOperatingConditions Instrument: PE SCIEXAPI 4000 BiomolecularMassAnalyzer SCIEXTurbolonSprayLiquid IntrodactionInterface HPSCLouCEmppugmen CPfDoArvSeometiPAtCroemomkptzaaxn)S1e31i106s0 Quatpamp GI311A pin py isees og Ble BNo4t0eL:7T40w0o) w4 ox t10amcmhiynpetrceaarfbedrrotph-inigpuasndvcaerterisdogesB(Koeystone,Lt# and/orHPLC system. -- nett 000163 | & | -- | D | | 1 | NICHonMojPbleiLcuoltCmieConPbnPoThlaeaVmussiopmelen(urA:lma)5te:u:,re:Gc23Se0ynMh.eCsiA esCy(Tm ones ACho creomsatteor gnrOapShyi o)l,2y.1Wm amtmerx 30 mum,dy. w3 ou%4 %B He03mali 37357s o00 111@00%00 5 00a03s33 5u o @ ,00533 pmeayrbienoeccsay adjust theHILC gradicat inonder tooptimize instrument Tap Appeosie POA Nepive UCPFOA Negative ga "23min 415-5370 ~2.8min. i2hbe1els0eern1piphotenehdcmcile.hesDmdcioyntothivuaiyn,lgiyohoonunogihdstaeyeoai-stcybeeapsia,pdeewliepaenp onthebs th of ivi ot: aaka LCIMSIMSsyste maybo usedonce demonstratedtobo 452. TineFlePramas 1 os com CO a) osA anTsom s0oo3leeutdL miofanosrotfsi hpePepFcorOiwzoAnocn(teeet1seoT0i.htmCusinoeendutfowreietnheiaallnkyyobnyesipndfduufsogiengeagp~mh1pga. s2a2d0a ng a4r3Ie3s,atvCedalt25teartcaunaiemnfPeirldeo.cTewhdiitrsetsun5e4le)iotfhecnaucsehdcduulrbienngtroonutinaeennaldysst. he Eames o Pst 000164 | & | L| . || D> i | ~~ S Ea ES O T . i pe sss toaa uesfor quan, nt Po Liverwandard cuherve ar ES E SEeE,nTE RT EE EE hE `statisticaloutlierbyusing outliertest (e.g. lest), T SErESorrS ea : 209925 (Z20.985). IFcalibrationresultsfalloutsidetheselimits, then <TT2 -- a Injectthesamealiquot (5iL) of each standard,sample, , control,etc. mSE EESmeEkmSE z e EA ter sampleset. In eithercas,calibration standardsmustbethe firstandJay ES EI rnc tT Ta E E n rR s `withinthestandardcurve range. ---- e Fortificationrecoveries falingwithin8510 115% (80to120% forlevelsat _--r e S -- rr e t co e---- 5 Samplesinwhich00peaks sredeta i.signal ntrio<3.1) he 000165 L & L || ? | || | | t(i1m0epspbbutwaherreelLesLsOtQhan=th10eplpobw)ewsitlclobnecreenptarratteidoan os f<1th0epcpabl.ibration standards meene 4.6.ACCEPTANCECRITERIA on Thefollowing criteriamustbemet toensure the presenceofPFOA and UC- 1. ToFnRoO: sutamts oaonst3ih0owstooe r lgloirne pes4t 13a 2. An"yC-sPFOeA: pesto mtd lak 2daughterionat370smufr om aparentof tbe tes 415amu 1dowe thn tfohledLlLowOeQr.thAanntyhaenLalLyOtQep.resentinthe reagent blankmustbe atleast5- 3B1eto5kn%rdw(nfaRu0ai21e0aioaonctr(ootiironccosonfsbooLpoLmltaetp losnfig.ySopnon ieeenvp315. ibe cioitte eptaol egelBOd ee ee 4 CpSnEyici3bae5ctsoofifchsadleinawnfyaosueasofbessesttsilsei eeolrrdeb7y mitr g8 1x1 BCU cnet mpm 0 to11n0 47 Peroncarn 5. TreeTesvaea e pe umentste i, T2he0com9e(la79t2io02n9c8o95e)f.fiIcifecnatlib)raftoiorncarleisburlatstifoanlcouruvseisdegtehneesraetLeidmimtsu,sttheben Thiem lovine igtomcofctesrssthbeephrwtorned myeasytttt,b,eor cdii4 nnS`ternsteeiofapn Foi aenit 2rSiioned1L0Q BogenResch Page or 000166 L& D | | | R`SuemcondsCeriotefrisotna:ndardsof iv ormorsconcentration levels,spamming a ange i`esngttarterehrtiisenaoignnoaantlsyomswriiebste.,hlsGoaewcpntoelhereftLcoLiaeOaytcQboaulefipbedrn1ae0lttityoheznecnehtudiwigrihoeetnshots(rce2gon)andccoaehnnf,dtsaraamtllioeonmslptaee0vn9enl8eot5so.bbGesirne3celuwndoced. 43. TomRaqTOuRAENiLEYEDS IpsAibsoocereatdtoaofrrsy3ic5nsoapompllrespsio(ke1sx,eaaidg8ah3tmoc0ounssatabomlypt,lae1m)emscpaalenbrxseyocnto.aknTeenhH,eoL1uOlagMbhoSrtaMthoSry.osopniaksa,on2s. (standards30035sample) willak spp 9ho: 5. CALCULATIONS 5.pUbesyaektBaqrAeuasa)oaunsyi1nsgfotofhtcewaalsrcteualpnardteaortgdhaecmsa.rovem(elionefasrraogyrosssfioounnpdariamdetenrs,)gbenaesreatoend oe Eautio1n; Analytefound(ppb)=(AssisPeak realocaksca) iteresg)x1Sconc. (ng/mL) b.EFqourastaimopnle2s0fcoratlicfuieldatweitthehpkrnoewan recovery. amountsofanalyteprior toextraction,use ReEcqouvaetriyo2(n:)= Analytefound(pp"bA)m=ovun3t.AAnnaslyytsefaodduerd (ty incontrol(ppb), x 100% 6. SAFETY ThIahangebneodrnaiatntnaosglryyscbsteotafnusodshrao,ersudlpsede0rcyeoarmrdleitaanhsggeesmt,tasht,oseirdnimgcaleldotisvhnaeogfsde.wtDoyrodUkasitsabne.gsIuhinneiefvtueosrmsfeaoolbrpaopedlrdslecspbutaeatsnniododanwrsocdsaweathkneesedg : Prowohean biandoingnsecsu. Exygen Research Pugs 150r20 000167 Jee RGettre | Table L RecoveryofPFOAfromFortificationsIn Monkey Serum Bp nm bm td Ried Skee T EomEmeRisaitc Lcaomovnnweoen sE Gmowe llbs 0%= amansAtAoDmpBypova x3% SummaryofPOARecover 10 ppbection okey eran Be me bee ae ied de mTmmy miay GR LuemEeoGTs ne meane = i 2 % mama sSoAuDEoben 5= Suey oPFOARecaro 100pp Bottini nMokeSor T Gr miTnRal men r oes w ~~ ma ecosup ws me 8 |> seAmnSTEAANBDAARDDEDEVVIAATRION: B2e ovina cvmace: " OVERALLKATIESona pA 2 | Boot Puetsorzo 000168 & er --------Ct" Figure1. CalibrationcurveforPFOAinControlMonkeySerum ' | : bmg | L / | orp Rech -| SPR eam Tine 000169 od Figur2e. Representative Chromatogramof a ControlMonkey Serum `Samplefor PFOA with ~ 5ng/mL of "C-PFOA Bl; EpE---------- ==. 5 Eis | | | | Rl | ET || . I! Bopatumss . Amin mm] Page 180120 000170 X @ | |Q :) | || | ||| ] Figure3. RepresentativeChromatogramof a PRO inConnMonkeySer ih EE- v pga.oC. =e | ' El= w=. BF: SH | Lad -. Page 190120 - 000171 | @ | | I |' | | | Figur4e.RepresentativeChromatogram of Control MonkeySerum Fortified at 10ppbwith PFOA andwith ~ 5ng/mLofC- PFOA E=- T Bi: A] Eat E=---e , i ' Jee AA. iic : =a ! ExygenResearch. Page200120 000172