Document 85MZg651vvdBGM1VRQRoOXojm

E. I. DU PONT DE NEMOURS & COMPANY KREBS PIGMENTS DEPARTMENT 256 YANDERPOOL STREET NEWARK. NEW JERSEY Library Fila TIT:; Ss NEWARK PLANT PIGMENT COLOR RESEARCH REPORT JACXSOH LABORATORY FIGMENTS GROUP RESEARCH REPORT PIGMTS FROM DERIVATIVES OF 2-AMIilO-BEliZOIC ACID (AHTHRANILIC ACID? AHD RELATED INTRRISEDI&TES Period Covered: February 3.1947 February 201948, FILE: DATE: 222,2 3/26/48 N42153 Njea7o Serial So. 101-48-4 Copy loo *3 1 - Sumerleal File 2 - Research File (222.2) 3 - Library File (222.2) 4 - Dr. JV E* BooWiXsi. 5 ~ Dr. !?, F. Spangoman*, Iswark 6 - Mr;, A* SXe^el/A.A.BrAesolara, iewark 7 - Br. D, B,, iCIXXian, Jackson lab.. Wito. 8 - Sr* A. D,, Reid laager, * 9 - Mr. Jo 1. 1 iakers * " 10 - Mr-o Jo Mo Sinker* t} 11 - Imperial Chemical Industries, ltd a 12 - " " K u (i 13 - 58 18 14 Extra Copy j a c k s o i ijmmmmi $mm$s mow r es ear c h r epo b 5?m.E PIGMiS FROM DERIVATIVES OF 2.4i09K~S8i20$C AC3 uifm&Miiic a c id ) m> musm ik t e b k b b ia x e s ... p e r io d CQFERJSB; February 3, 194? to February 20, 1948. CEftBOE* A-II-C-238 SUBMITTED Sis A* ,D. Bald ingel* APPROVED Bis Do S, Killian BAKE SUBMITTEDs DATE ISSOEDz DUP050066906 Investigation was mads of the usefulness as .-dla&o components of a number of Intermediates related structurally to 2~amino teensoic acid (antfaranillc acid), Sam of these'had teen evaluated a number of: years ago and la. view of tha results- than obtained-, further study appeared to be warranted. As a bos is for comp.ariso;nf couplings of sntlaranilic acid to various second components war used, Improvements In the hake Bad D type pignssit (anthranflic Acid---> Beta Baphthcl) anil In Pigment Scarlet take (aiithruailie Acid H-Salt) Yfere looked for. It was also planned to check earlier work "which* Indicated that pigment of "fhtdiung1* Rod shads (Permanent Red 28 Acid BQtO could he obtained from derivatives of anthranilic acid or their isomers. mmmumsasmsm Of the intermediates tried, 4chlar2-sm.ino `benzoic acid appears to be of most Interest., Iho manganese' salt of the coupling io" BOH was a maroon pigment somewhat lighter' than (?OB**ii> BOKj Mr) with much yellower undertone. It m&y have application in automotive enamels,particularly In metallic finishes .In .which PUS #143), the K-25X2 formula is attfeetesd,. k sample <18-14-4) representing the manganese salt of -S-eb-tor2-amino tes.nko.ic acid-^ BOf? was also prepared for evaluation, Bills is a maroon about equal In depth to Ef-533-B {JPCASBA---^ B01) end therefore lighter than tha 4~etelsr derivative, it is of- interest tee cense the interned late cm tee made from, a cheap by-product .of the Chambers Works 6ctelor~2-ait3rotoluene. A close tinctorial taatch for ^Watchung** Eedj 8$-428*4> was obtained from 2-chlor-!?'-amino teen&ole acid coupled to 801 (Ca 'salt}? provided the color was' flushed into varnish-, fte dried toner wa& weak. fteis interne-late is at present too expensive for considera tion. P-amlno turnsole acid coupled to SOI? also approximated the . -rfatchungs Rod shade. Ifee higher -cost of this Intermediate compared-' to Rod .3 sold would make its .use uneconomic* imlnoterepfatte&Xte acid coupled to Bata laphtliol <Ca salt) may tea of interest as ah Intermediate for a .Bake Bod R typo pig ment. Bis product doss not show the sensitivity to drier' eafciteited by Lake Bad R but on the otter -hand hm poorer 1 ightfas tness DUP050066907 \ 2w msmmj&jmmx --Tbs lln salt is described above* The Ca mas similar in shads but duller and less lightfabt* 'T^Beta faphthol, The Ba salt showed no advantage over taka Bad J> The product *** somewhat yellower and mealier and exhibited the characteristic sensitivity to metallic drier* E-Salt Ih the tom of Pigment Scarlet Lakea of RL~211~D type* the products obtained wars hard la texture and weak in tinting strength* Pulps of barium sM strontium toners, tested by paper dyeings, showed no advantage over Pigment Scarlet in strength or in lightfastaass* In the form of paper coatings <brusho.ut) the strontium toner exhibited excellent light resistance* BOI The manganese salt is a dull maroon of no interest* ^is product is similar to that from the 4chlor isomer*' --> W 'The Ba salt is a strong clear-tinted yellow possessing very poor lightfes.tneas* . ' The Ma* salt is discus sad in the Summary* This product'exhibited instability in ths making formula and also in the enamel from it, which turned brown on aging* Development of the color at 80C. instead . of at a boil gave more consistent results* The Ca salt, propped by a rosin&ted formula, is a dark transparent reel possessing excellent baking and bleed resistance* BOH The Co salt is close to 3hfe.tclmag^ Bod, BT*428~J>, in -shad and if flushed from the filter cake Into varnish is equal in strength* Drying the color re* suited in a hard, weak pigment* Lightfs-stness and bleed properties' were inferior to the ?kfatchung!* colors*' DUP050066908 Beta Maphthoi, Ba and Ca salts had mors Intens a mas stones , and less bronzy finish than the corresponding anthranilic acid-***#* .BS pigments hut wens weaker due pre sumably to poor texture of the dry color* --*> PIP The Ba salt is a reddish shade yellow of fair lightfastness* fhe combination is probably too expensive to merit consideration* B1 Barium end calcium salts slightly weaker- than obtained from.the hasulforated intermediate,, Otherwise similar* ,,^ap go! Calcium salt was mak as a dry color with sosnwhat poorer .strength but more intense ass stone than the unsulfonatod intermediate* *:$* H-Salt Barium lake of R1-2XI-I3 type was hard textured and weak in tinting strength* *& BOS The calcium salt is considerably yellower in shads than `slatchungsi> Bod Toner, HT-428-D, is slightly worse in ligbtfustness sad definitely inferior in Mood pro perties. Texture of the dried product was good* The higher cost of this intermediate compared to Bed 2B leid would make its use uneconomic* *"> PIP --^ .BS *--> BOB Both Ba and Ca salts are very m&k yellom$ approxi mating Bensidins 'fellow %T~4$9~D in shade. The Ca toner is lighter and stronger than the Be salt and show a definite advantage in lightfestncss over 1T-459-B, its poor tinting strength would be & 'handicap to its pr(motion. The 2a salt is a weak red of no interest* The Ca salt is superior tlnctorlaXly and although somewhat bluer in tint may he of: interest as a lake Bed type. It appears to be less sensitive to metallic driers than the latter pigment tut ia not as good la lightfasIncss* The coupled dye mm -completely soluble as' the soda salt and was .not converted to *tfe .metal salts. DUP050066909 E&phthol* 3*ha product of this combination is an orange somewhat yallovyer then Parra* tone Orange, 12~419<D in shade with excellent lighifastnoss of'fall etrhagta d?8%Mioe PSl? A reddish yollow much wcak-iar tb&a the .strong tjpm BssizMlaa fellow, '12*553-$ with about equal lightfastaess, 'Bi&sotisation of this iuterstedicto was effected by ass of aitrosyl sulphuric acM Since' coupling did mt taka plac^ readily In acid solution, neutralisation of the --eacess acid was necessary# As the 5-ehlor derivative is soluble ia - hydrochloric eeid solution, it mj he possible to develop a hotter method for disaotisatioa* -*f Bate Haphthol.* in orange si.Hr.:' to Orange 02 (BOA- JAA.P) in shade hut considerably weaker* ifio difficult-/- of die'sotisfe.g am coupling mzf account for the lack of strength and also ths poor llghtfastncoa which eras obtained* ^EtoenyX Bffisthjl fyuagolonse A reddish yellow similar to that from the f-ehlor derivative Mt considerably weaker,. Ss.2L.lliei:iaii:ilAa,.Mis, A deep maroon ^igaont. ecnHderebly bluer than Am Bordscu:t lake, ES*'3$*B? aM superior in lightfustacwa* Because of hard texture of tho"dry color, evaluation t o * mads by flushing from'the rater paste* fhe coMbinatioBs tasted aau the corresponding notebook references arc listed belows. - l-|ihayl3*jS0tb.yl*5-PiP,^^o3hh ***a^ Beta l&phthol **P> Beta oscy aaplathoic acid te^8, IB 1234 n libspt, 4 16, 21 . 22 18, 25 36.# 51 DUP050066910 2*ejaino-g4-chl&g bsmolc ac Id -h ? son **$> 'B*SXfc .2S*Wk< "**g* BOH w&H-Salt ESxplJp 4 '5? Expt422 18, 25, 2? 12 . IB X236s ExpU 4, 58 " 285 42 ,f 19* 25*27> 31 11 36, 51 m -1260, gxpt.15, 24 , 35, 40, 48 j- 53 , IIS 1279V 8*t* 9, 14, 35, 46 ~g> BI IvCpto 4, 56 ffl&pt022* 48 25, 27, 31 2ehlo5Vana lno4~aulfo benzoic sold BIT *$> BOH R-Salt IB 1si23.6 ?s Exptp 22, 42 Bxpta 19 Bxpt.o 12, 36 Jfcfiffll >,gGQ.a.d.c Acid IB 1236 , %xpU 2?, 31 IB 1236, Mxpti 53 st DUP050066911 ** & TO i 33 30 47 Eapt* 50 SOM 5*5i **& B-Salt IB S^pt* 33 Bn>t 30* 47 SxpS* 50 SB .X2?9?. Expt.. 30 Attached Is the foamXn foy tha preparation of R25>12 (4~chloy-2-a&iao bimaoic aoid-^BOlij, Ita). SJti-a d*ehlor derivative ms a&de fei .simiXcir^iaamies? asjeepfc that It was developed at 80C instead pf at boil* DUP050066912 ..->5 .-% r ? (. . i . ;i >. . .. . . , -V i . ... V `;| v: D.r.44i ^ lf;43 V.t ,'::'av* i?$,r izzrr z^zrirzrrr^^iTrir ...a r-nv-T ->y '" ?~ - . _..J'ililv. ..... ,, i sift S:"'. | s. L:r.;-..i... . ? 2-u&ii<s 'Sadv-s '2.00$ j______ 'j_ 44 1 JOO 52^GO ul* :g|j5r.t. usli ofrPfh Iv ,253. _Jkf2 * " tsIF 1.0# ^*yly 1CH20 j,iaat ar, r in, c :*.g;.'?!? t, ' cats_sli.VjVj. ^'r\ :.~-j ~Viw v _32 Z/Ji^ _v _n___ , ._.J: ***, ____ ____________j 30 j iJO .c'i^lvsa aa -aoM h Is f *.... ........_ _____ L.,-___.j____ . &#r-v$$r,....... _____ _____ ______L~___ J,,j1 Ov-it-n In g,s O'-t r: .o'xirXbls__ "T.r^."..i.. '..."...(.. ~ 0B*f | 1C> -Mrueat), 5? m 44 ..400 j 4____ ISasseis*. i'fo J-M... j&ggSLJ ril^s&agLS^I fenaiis jia>< 1P(4,, ; 44 f j|.. 7 ,, J* \ i.) ~ _ UCA iQ $?$_'*___________ ___________ _ ~r' ........ ..... * '' 5iZiEil;M,,.JJCIj l ........_________________I to 4l3.s.Go.?.vg., r.JS:iksL.3M__________ _....._______ __JL i____ 3 J*?. !. ;,r044...s.c.;.4 ;tot^.. ms.3 Sofka -da-i 1 ' "T i ! ' 1 f ?5 ;r625 T.rtor m X$$-*).0*W ! 1 .1 1 . 1 ! : Ocwale. iisjas 00J sokrtim 3 1 i tin 30*40 t&stxazt Bf thru etii 'feuetlc J&0&-.9 100/i ' '{*#* S(d r.-im ?3 1 40 ! f eo^l^g) Jt ,mc3- bz f aid. (Final Urtt . 801^,515.6 -JUf JOS .Salt l 1 .. . t ........................... -...... r "... ' fi'OAt. TlfK-S1., rras- i I ! disaolTsu in I 1230 i 10S.G# eo3,i oc.isr . .. !!! S' \. 1 1 (Test riltrat sligrlt oa'33 I 11 11 Eeslarry ii3.isir oeke in' J 3Q0D ! 25000 | . J'. 1 . . : ..'...... :.......-..:...........r'. 1 _ _ _ _ . . ... f,, ,-COCT -S~0"?_ DUP050066913 ......... ; " ; CXV'iiC-s^,^_ __...,,_____ ' vy * .`c:;-;; '.y'y t ? i j 'I' * ' " ^ 2 s` - Tcass? V t> m- astt s':;. ......rI :xv;:a.-; 1 \M SO ; 3-g5 _ ' oc?.fl sy &1Z1.1 __ jjjt "i"w fafo ~ s:.3>*UrV ' S--------------- ...' -~^lr gOO i -s X$ .Mcl >4 Is^lg iAsaisiS __ J j Sl . OSl . &t** t \ \ _.......................... f .. ----- ! ' --. ...... tc ->B Y * & f 83 _____ is. 5I T~~' I Via ________________ ___ ..io ..J_______J'.........................MMMil. .... . ! u p^ls^si to V ?.5v0 : f^s^a.riiisasPe ,........................ __ ____ _. .,.................,, ..- *i 1 .............................. .; 3 3 ! - ::a5a?i 1 (r^ssiU ;gl{ -..T<4).................,,....... . ' ....................... ... 1 i. at ;,40!:'fo 1-___ L____U- niOtwr.lye 11 i__ J X.... "* <v i_,,_J 31 J. 1 \ 1 . r ............. 11 r' ___ L________ . > . J_ !. . L .: . r '................... ..... . *... ...p ... x........ . . . ' i: . .A ' . .. 1 ! ......... .. " r .!'; * ........................ i' i r*J 1 fAWJS-~lSi.--- MBS. 'FWi-JSOS--. .......... ...-............ ....... ... ifl-ifl ~i r": : '! -V. *' cr- j g p&? immm. JL .jKsramjSsKU &, ,, sEmiioasR'^t^*' DUP050066914 wmjmisim XhJ# :imrQim ia W jfoilO# TO&ertooe .esc! ii;at in raisiios to sasstO:a&>, 'tho festayla is tesofi an pm^e&vtmn ttf*o$ fw sisalier piggteKrts m& ii^ormtioa t o o Sstsdaed 9.6 to -sfre^i e? TOrl&Xjr* Cesii>Xt iiaerli miles of aoEt&rsjsilio id $m sow iiffiaeiij fie. to tli* low s0lat3lIi.iT of its hy^tooSdoviM* 5I* effect of a loag^r stirring perlcfi t o o 4fc*tfJdU Cmiplisg i.a papoooaoo of eofiiem oariHmafce prmzmIn m-ddf if the pB is mieiair^.d sfep ?&* Mfiitioa of osairiio scia lasjr feo '&6* if aoooMiay# Xs3latlo of if** %& s r t o & 4os&r 'oluor product ifes ufcfcn &&s*:rict otrol^rt ttira* -."t 'a gs$s&bX to saroifi with salt .s o '&j v Io b. bp ad^uotoamt of pf alien soapliag to a'ouut 0,0* BEJJWi:eSmE. ' \ 3/19/ .CC DUP050066915