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CORNING Hazleton MUTAGENICITY TEST ON T-6342 IN AN IN VIVO MOUSE MICRONUCLEUS ASSAY + [EINALREPORT AUTHOR Hemalatha Murli, Ph.D. PERFORMINGLABORATORY Corning Hazleton Inc. (CHV) Vi9en2n0a0,LVeiersgbiunirag P2i2k1e82 BE : ; CHV Study No.: 17073-0-455 SUBMITTTEDO 3M Corporation SBt.uiPladuiln,gM2i2n0n-e2sEo-t0a2,5351M44C-e1nt0e0r0 STUDYCOMPLETIONDATE December 14, 1995 CHV Study No.: 17073-0-455 1of23 00330 CORNING Hazleton QUALITY ASSURANCE STATEMENT Project Title: In ivo Mouse Micronucleus Assay Project No.: 20996 Assay No: 17073 Protocol No.: 455. Edition No.: 17, Modified for 3M Corporation pQruoajleicttywAesrseurcaonncdeucitnesdpeacctcioorndsoinfgthtoetshteudSytaannddarrdevOipeewroatfitnhgePfrioncaledruerpeosrotoftfhtheeQaubaloivteyrAesfseurernacnecde rUengiutlaatnidonasc.coFridnidnigngtso tfhreomgetnheerailnsrpeeqcutiiroenmseanntdsoffitnahlereappoprrtoprreivaiteewGwoeorde Lraebpoorrtaetdortoy mPraancatgiceement and to the study director on the following dates: RandomizationofAnimals/09/18/1995 Draft report Review/10/31/1995 Final Report Review/12/14/1995 09/18/1995 10/31/1995 12/14/1995 S. Ballenger C. Orantes C. Orantes Quality Assurance Unit 12/7 4 DaeReltased CHV Study No.: 17073-0455 2 G00331 CORNING Hazleton STUDY COMPLIANCE AND CERTIFICATION RaTsehgesueltdaeftsoicrortnihsbiePndatrshtteu5Fd8oy,owidsassaunecddonDDderucucegtmeAbddemirinn2ci2os,mtpr1al9ti7ia8on,nc(e(efFwfDieAtc)hti,tvheTeiJtGuloneeo21d2o0fL,at1bh9oe7r9aU)t.oSwr.iytCPhroaadncetyoiacfpepFrleedgeurlaaltions saimgenneddmpernottso.colThtehartewwoeurlednaoffseicgtnitfhieciannttedgerviityaotifotnhsefsrtoumdythoeratfhoerienmteenrtpireotnaetdiorneogfutlahteiotnessitcorarebstluhelets. tTehstearratiwcldeaatsa hpraevseenbteeednhreerveiienwreedprbeysetnhtesSatnuadpypDriorpercitaotre,cwohncolucseritoinfiweistthhiant tthhee ceovnatleuxattoiofntohftehe study design and evaluation criteria. rAelclotredsthaasndbecoenntrroelvireeswueldtsbiyntthheisSrteupdoyrtDiarreectsourp.poArltledrabwy daantae,xpdeorciummeennttaaltidoant,a rreeccoorrddsa,npdrtohtioscol faancdilaitceospoyfofCotrhneinfignaHlazrelpeotrotngIennce.rfaotredatalseaasrtesounletoyfeatrhifsolsltouwdiynwgislubbmeisasrcihoinvoefdtihnetfhienaSltorreagpeo.rt to mattithmeeerS,ipoaorlnsssoerrnet.ttai0Anfeatdesrtiontrhtaehgeoensfetaocyirleaigaterypfdaeecrsiiilogidnt,easttheoedfSbCpyoomtnhsieonrSgpmoHanasyzolree.lteocnt Itnoc.hafvoer athneaadfdoitrieomneanltpieornieodd of Submitted By: Study Director: Hemalatha Murli, Ph.D. DMeapmamratlmienatnoCfyGteongeetneitciacsnd Cellular Toxicology Study Completion Date CHV Study No.: 17073-0455 3 00332 TAOFBCOL NTEE NTS CORNINGHazleton SUMMARY iii 10 SPONSOR oot Page No. 6 20 2M1 ATECl(iTeeR nts'tsI AIrdteincAtlief)iLcation .......................oooo..............7 22 DateReceived 23 Physical Description 24 Genetics Assay No. 30 TYPEOFASSAY............ccooooiiiiiiiiiiii 40 PROTOCOLNO............ccooiiiiiiiiiiiiiiiiiiiiiiiii iT 50 5S1TUDYDAITnEitSia.ti.o.n.D.a.t.e...o.oooiiiiiiiiiiiiiiiiiiiiiiiiiiiiiiiii il 52 Experimental Start Date: 53 Experimental Termination Date 60 SUPERVISORY PERSONNEL 61 Study Director ................ccccocoooiiuiiiiiil,..7 62 Laboratory Supervisor 70 OBJECTIVE ......ooiiiiiiiiiiiiiiiiiiiiiiiiieeeeee eT 80 MATERIALS ............................. veverssronnnis 90 SOLUBANIDLSTAIBITLITYY: ..............ccccoieee iii 8 100 DOSE SELECSTTUIDYON 10.1 DoseSelection ..............ccccciiunneniiniiiniinnnnill 8 102 Dosing Information 103 104 Results and Interpretation Conclusion CHV Study No.: 17073-0455 4 00333 CORNINGHazleton 11.0 M111ICDRoseOSeNleScTtUiUoDnCY.L...E...U..S....ccccveeeeeenseiiiiiiienn. 10 12 Micronucleus Assay Dosing Information 120 BONEMARROWHARVEST,SLIDE PREPARATIONANDANALYSIS .....11 130 EVALUATION CRITERIA 13.1 General ................ccccceiiiiiiiiiiiiiiii 12 132 Data Presentation and Interpretation 140 RESULTSANDINTERPRETATION ....................................13 150 CONCLUSION .............ooiiiiiiiiiiiiiiiiiiiininnnnn 13 160 REFERENCES.................cooiiiiiiiiiiiiiiiiiiiiiii 14 170 EXPERIMENTDATATABLES ...................ccccceeiiiiiii1ii5i CHV Study No.: 17073-0455 5 00334 SUMMARY CORNINGHazleton Mutagenicity Test on T-6342 in an In Vivo Mouse Micronucleus Assay `The objective of this in vivo. assay was to evaluate the abilityofthe test article, T-6342, `micronuclei in bone marrow polychromatic erythrocytesof Crl:CD-1%(ICR) BR mice. to induce In the dose selection gavage at 500, 1625, study,thetest article was solubilized in deionized water and 2750, 3875, and 5000 mg/kg. Six animals (three males and dosed by oral swiegrnes aasnsdi/gonremdotrotaelaicthy d. ose group. Animals were observed for three days after dostihnregeffoermatolxeisc) >B5as0e0d0 omng/tkhge.reIsunltthseofmtihcreonduocsleesuesleacstsiaoyn,`tshtuedyt,estthaertmiaclxeiwmausmsotloulbeirlaitzeedddionsedewiaonsiezsetdiwmaatteerdaasnd dosed by oral gavage at were randomly assigned t1o25e0a,ch25d0o0s,e/ahnadrv5e0st00ti`mmeg/gkrgo.upT.enVeahniicmlaelsan(dfipvoesmiatilvees and fivfeemales) control groups euthanatized with the test aarptipcrloexwiemraeteeluyth2a4nahtoiuzresdaafpteprrodxoismiantgewleyr2e4,in4c8luadnedd in 72 the assay. The animals hours after. dosing for dosed extraction ofthe bone marrow. `The test material, T-6342, did not inducae significant increase in micronuclei in bone marrow polychromatic erythrocytes under the conditionsofthis `mouse bone marrow micronucleus test. assay and is considered negative in the CHV Study No.: 17073-0-455 6 G00335 : CORNING Hazleton Mutagenicity Test on T-6342 in an in vivo Mouse Micronucleus Assay 1.0 SPONSOR: 3M Corporation 20 MATERIAL (Test Article) 21 Client's Identification: T-6342 22 Date Received: July 21, 1995 23 Physical Description: Clear, colorless liquid 24 Genetics Assay No.: 17073 30 TYPEOF ASSAY: In Vivo Mouse Micronucleus Assay 40 PROTOCOL NO.: 455, Edition 17, Modified for 3M Corporation 50 STUDY DATES 5.1 Initiation Date: August 15, 1995 5.2 Experimental Start Date: August 29, 1995 5.3 Experimental Termination Date: October 16,1995 60 SUPERVISORY PERSONNEL 6.1 Study Director: Hemalatha Murli, Ph.D. 6.2 Laboratory Supervisor: Monica Vegarra, B.S. 70 OBJECTIVE i`TnhdeucoebjmeicctriovenuofctlheiisininbovniveomaasrsrayowwapsoltyocehvraolmuaattiectehreyatbhirloictyytoefsothfeCtrels:tCaDr-t|ic1l%e,(ITC-R6)34B2R, to mice. This study was Heddleet al. (1983). conducted `using modificationsof the procedures suggested by CHV Study No.: 17073-0-455 7 G00336 80 MATERIALS `CORNING Hazleton mRAiadvuxelirtmiLmzaabeloergaeatnnoerdtiifecse,hmeaPtloeerrtomagigecenee,MiLst.ty.raainTndhCiarstlht:ehCaeDls-th1ay%m,(eIrtCaiRnm)deoBamRs,sburwreeedrasectcrpeauisrnscwhtaoassaescdeolfemrcomtmoednChtsoarles dTohseinpgr.otocol for this study was approved by the CHV-ACUC pritoothre initiationouorfce. c7Aa2ng4ie6maaltFsraawnndedro5mei5zhao1tu5isoe%nd.ruepsTtpheoectsitevevemlepyne.rpaeAtrucr1ea2ga-ehnodduurrreillnaigtgihqvtue/a1hr2ua-mnhtioiduniret,dyaarwnkedrcheyocmulaesiewndtaauipnetod fative per aAvaciolmabmleercaidallibdiitetum(PfuorritnhaedCuerrattiifoineodfLtahbeorsattuodyr.y PTehlleetfseed#w5a0s02a)naalnydzewdatbseyrmtawhieenrteained. rhmeyatdnrruoofscapacerctbtuiorvneesr,bfaoosrrigscaonfnoocrpehsnoptesrcpaihtfaiiotenedsso,mfiascpnredocosirpfgeiaceniidfishemedsa,nvupytersmiteeintctaisld.se,sT,ahfaellakwtaoalxitinenir,tywc,hahlseoraainnaaltyezded on a ahnaliomgaelnss.or Swaonriktiinzegdwciatghiinngtwheasanuismeadl ffoarcihloituiseisnwgertheeraeniqmuailsr.etodPewresaornnseuiltahbavlnyedlmpireonttagelcst,ivaen.d `garments and equipment. arAnaninimdmaoalmlslsywweaersreseidgqonuseaedrdatnbotaissnteeudddyufpogorrnosuetpvhsenainnbddeifwvoeirdreueableiinbdnoigdvpiyldauwaceleilgdyhotwnse.sitgAuhndeyid.mapArlnisoirwmeatorlesdouwsneiinrqge.uelAyll identified by ear tag. Dose or treatment groups were identified by cage card/label, iAnthatlhaetitoenr,mifnoaltlioownedoftbhyepesnteutdryataillonosufrtvihveintghoarnaix.malAsnwyeerxetreautahnainmaatliszendotbyusCeOd,for the study were cuthanatized by CO, inhalation, followed by penetrationofthe thorax. 90 SOLUBILITY AND STABILITY: The this atsesstayarwtiacsle,deTi-o6n3i4z2e,d wwaatsers.uppTlhieedstaasbialictlyoeafrtchoelotrelsetssmaltieqruiida.l uTnhdeervethhiecldeossienlgected for conditionsofthis assay is the responsibilityofthe sponsor. 10.0 DOSE SELECTION STUDY 10.1 Dose Selection `Dgoasveagelefvoelrstohfe d5o00s,e s1e6l2e5c,ti2o7n50st,ud3y8.75, and 5000 mg/kgwereadministered by oral CHV Study No.: 17073-0-455 8 00337 CORNING Hazleton 102 Dosing Information wa`eTnihdgeh2a1tn.ri1amna-gl2es5o.u1fstegdhraeimntsah,niefmdoaorlstsheseuesmleaedlcietnsitohanenddaosfsseaemyawlreeasrn,geerdeofsispneedcditniovgnealysA.suagyuDoswstais2n92g,6s.1o59l9u-5t3.i3o.nT5she `swteorcekfporretphareedhijguhstdporsieor(5to00d0osmign/gkga)n.d wTehrise pwraespparreedpabryedmbay akddi2inn5g0g60.6mgm/lmolf cdleeiaorn,iczoeldorwlaetsesrso(lLuottio#n.17,Dpirluetpiaornesd oafttChiHsVs)totcok6w.e0r0e07prgoepfarTe-d63f4or2,threeostuhletirndgoisn ea levels wDeoeskinsganwdasonaechdiaeyveodldusaitntghea t1i0mmeol/fkdgosdionsgi.ngAvnolouumteli.neAolfltahneimdaolssinwgersechceigmhetis found in the following table. A totalof 30 animals was used in this assay. TREATMEDNOTSE GROUPS MF T-6342 500 mg/kg 1625 mg/kg 2750 mg/kg 3875 mgkg 5000 mg/kg 303 303 303 303 ER All doses given were on an acute (one-time only) bass. 103 Results and Interpretation sAtludayn(itmharlese wdeayrse)efxoarmtionxiecdeafffteecrtsdoasnidn/goranmodrtdaaliiltyietsh.roAulglhaonuitmtahlesdauprapteiaorneodfthe onbosremravlatiimomnepdeiraitode.lyTahfteermodrotsailnigtyanddatraefmoaritnheids ahsesaalythayreunstiulmtmhaerieznedodfitnhtehe following table: CHV Study No.: 17073-0455 9 00338 CORNINGHazleton SuimnmMaircyeoDfosMeordtAacliuttieelsyWwiitthhiTn-363D4a2ys Observations 500 mg/kg 1625 mg/kg 2750 mg/kg 3875 mg/kg 5000 mg/kg -_-- 104 Conclusion 03 3 03 3 3 03 03 3 3 03 OOO Based >5000 on these mg/kg. results, the maximum tolerated dosewas estimated to be 11.0 MICRONUCLEUS STUDY 111 Dose Selection 5B0a0s0edmogn/krgewsuelrtsesferloemcttehde dose selection for this study. study, dose levels of 1250, 2500, and 11.2 Micronucleus Assay Dosing Information CTyhcelaonpihmoaslpshuasmeiddein(tShiegmmai,crLoontuc#l4eu3sH0a2s6sa9y,wCeArSe d#os6e0d55o-n19S-e2p),tetmhbeepros1i9t,iv1e995. cwoanstraodlm,iwniesstseorleudbiblyizoerdalignasvteargieleadtei8o0nmigz/ekdg.watTehre(Lvoethi#c1l7e,cpornterpoalr,eddeaitonCiHzVed) and amwriatctirecolren(uaLtcolate#uvso1la7us,mspaeryeowpfaa1rs0ed2m8la./t7kCg-.H3V7)T.,h6ewgawaesnidagdh2mt1i.rn1aisn-tg2ee5or.fe6td hgcoegnrcaaunmrirsmeafnlotsrlyutshweeidmthailntehtseheatensdt amfdeadmkaiilnneggs,daeri5eos0np0iezcmtegidv/ewmlaylt.esrtTothcoek1fd1oo.rs0it0hn0eg8hsgiooglfhuTtd-ioo6ns3se4f(o25r0ut0ph0etmoagsa/skavgyo)lw.uermTeehoipsrewpaasrepdrebpyared by tchleearr,emcaolionrilnegssdososleutlievoenlsw.as obiained. Dilutionsofthis stock wefre22p.r0epmalr,edAfor CHV Study No.: 17073-0455 10 G00339 CORNING Hazleton hTaernveasntitmiamles g(rfiovuep.malVeehsiacnlde afinvdepfoesmiatlievse)cwonetrreolragnroduopmsl,yeaustshiagnnaetdizteodeach dose/- dapopsreodxwiimtahtetlhye 2te4sthoarutrisclaefwteerrdeoesuitnhga,nwaetrizeeidnacplpurdoexdiimnattheelyas2s4a,y.48Tahneda7n2imhaolusrs after dosing for extraction ofthe is found in the following table: bone marrow. An outlineofthe dosing scheme. Dosing Scheme for Micronucleus Assay A totalof 110 animals was used in this assay NumberofAnimals Assigned Treatment eZ 1250 mg/kg 2500 mg/kg 5000 mg/kg Vehicle Control, dei1o0nimzeidgwater _P--ositive Control, Cyclophosphamide, 80mghkg 2M4FH 4M8FHr TM2HFr 55 55 55 55 55 55 55 55 5s 55... 55 - - - - TVhoeluamgee odfostehde awnaisma1l0smalt/tkhge atnidmewofadsobsaisnedguwpaosneiingdhitvwideueaklsaannidmaolnweediagyh.t, 120 BONE MARROW HARVEST, SLIDE PREPARATION AND ANALYSIS pAetnetthreaatpipornoofprtihateethhaorrvaexstantdimteh,etahdehaenriimnaglosfwtetriesseuuethaanndateipziepdhywsietshoCfOb,otfholfleomwoerdabwyere croenmtoaviendi.ngT3h-e5mamlrrboowviwnaessfelruusmhe(donferotmubtehefobroenaechanadnitmraaln)s.ferFroeldltoowicenngtrciefnutgreiftuugbaetsion to pweelrleetstphreeatidssoune,sltihdeessuapnedmaaitradnrtiewda.sTrheemoslvieddesbwyearsepifriaxteidoninamnedtphoarntoilo,nsanofdthsteaipneeldleitn cMoavye-rGslriupnpweadludsisnogluDteiopnexfolmloouwnedtibnygGmieedmisuam.(Schmid, 1975). The air-dried slides were eTrhyethsrloicdyetsew(ePrCeEc)odtoednofromroacnahlryosmisa,tiacndersyctohrreodcyftoer (miNcCrEo)nuccelleliraatniod.thSetapnodlayrcdhrfoomramtsicwere CHV Study No.: 17073-0455 n 00340 CORNING Hazleton mPuCisEceSrdsotnpourcreleseceaonrttdeidtnhcteehlselessdwcaoatars.edeOxopnpreteisctshfeoideulsda.asnpdTehrPecCeEnntoSrmpmieacrlraofnnriuecmqlaueleanwtceeyrdoecfesmlciloscrrebodan.suecTdlhoeeinfitrheeqtuoetnacly of Crl:CD-1%(ICR) BR strain is about 0.0-0.4%. n this TNhCeESfroebqsueernvceydofinPtChEesopvteircsfuiselNdCsEwhsilweasscdoertienrgmtihneedfirbsyt 1sc0o0r0eirnygtthhreoncyutmebse,r of PCEs and 13.0 EVALUATION CRITERIA: 13.1 General MTihcerocrniutcelreiaifwoerrtehedairdkelntyifsitcaaitnieodnoafndmigcernoenruaclllyeirowuenrde, tahlotsheooufghSaclhmmoindd(a1n9d76) rainndgwshearpeegdemniercarlolnyucbleetiwoececnas1i/o2n0alalnydo1c/c5urtrheeds.izMeoicfrtohneucPlCeEi.haTdhsehaurniptobfosrdceorrsing mwoarsethtehamnicornoenumcilceraotneudclceeluls, nwoatstchoeumnitcerdoansucolneeusm;ictrhounsutchleeaotcceadsiPoCnEa,l ncoetlltwwioth(or more) micronuclei. of PCEs and NCEs (Tbhleuisstha-ignrienyg apnrdocreeddu,rreesppeercmtiivtetleyd).the differentiation by color 13.2 Data Presentation and Interpretation DInadtiaviadrueasluamnmiamrailzdeadtabyarseeaxlsaondprdesoesnetegdr.oupTshefoarnatlhyesdiisfoffetrhenetsteimdeatpaoiwnatss. p(ewrhfeonrmvaerdiaunsciensg aarneahnoamlyosgiesonefovuasr)iaanncder(aWniknetrr,an1s9f7o1r)meodn(ewihtheenr uvanrtiraanncsefsoarrmeed hofetvearroigaennceeowuas)s psriogpnoifritciaonntso(fpc<e0.l0l5s),wiatDhumnincertot'nsuctlteeistpe(rDuannniemtatl,. I19f5t5h;e 1a9n6a4l)yswias s unesgeadttiovedceotnetrromli.ne Awnhailcyhsedsosweergeropueprsf,ioframneyd,sewpearreatseilgyniffoirceanatclhy hdairfvfeesretnttifmreoamntdhe ssteaxticsotimcbailnlaytsiiognni.fiTcahnet cdroistee-riraelfaotreddeitnecrrmeiansienignamipocsriotniuvcelreeastpeodnPsCeEiSn,voolrvethdea dleeatsetctoinoen doosfaerleepverlo.duAcibtelset aanrtdicslteattihsatticianldlyucseigdnnifeiictanhteaprosstiattiivsetircealslpyonsisgeniffoircaatnt dleovseel rweasspocnosnesindoeraredstnaetgiasttiivcea.llyIsnigeniitfhiecracnatsae,ndthreepfirnoadlucdiebcliesiionncrweaassebaatseodneondose scientific judgment. CHV Study No.: 17073-0455 2 00341 140 RESULTS AND INTERPRETATION: CORNINGHazleton adAunlrldaaptnoisioinmtaoilvfsetwcheoenratesrsooalbysgefrroorvueptdosxiaimcpmpseeydaimrapetdteonlmoysramafatnledra/fodtroesmrionrdtgoaslaiinntdgiepsae.nrdiAordleimcaaanliilnymeadtlhshreoianulgtthhhoeyutvuenthhiecle aappppreoaprreidatneorhamravlesitmmteimdeisa.teAllylaatneirmadlossifnrgoamntdhere1m2a5i0neadndhe2a5l0t0hymngi/klgtdhoesaeppgrroopurpitsaitlethe harvest times. Immediately after dosing, all animals in the 5000 mg/kg dose group appeared normal, hAopuprrohxairmveasttelgyro2u4p)hofurrosmatfhteer5d0o0s0inmgg,/2kgmadloesse(g#r'o52u7p1w2,er4e8fhoouunrdhdaeravde.stOgnroeump;al2e714, 72. a(n#i2m7a1l8s, a7p2pheoaurerdhanrovremsatlgratoutphi)satpipmee.ared hunched and weak with squinted eyes. All other fAepmparloexi(m#a2t7e80l,y 7428 hhoouurrshaafrtveerstdogsrionugp,)|fmraolmet(he2751080,0 7m2g/hkogurdohsaervgerstougprowuepr)eafnodun1d dead. Al otheranimals harvest times. appeared normal at this time and remained healthy until the appropriate opTrohleaytctaehnsrtyooamfratttichilcee,ehrTay-rt6vh3er4sot2c,yttiiemnsedsou.vceeDrdutnhtoeoslietgvonexilifsciicotabyn,stetrihnvecerPdeCaiEsne/tshNeiCnvEmeihrciacrtloieonsuoccoflntetrahotelesdmailn eesitahnerd sex lfoewmearletshafnrotmhethveeh5i0cl0e0cmognt/rkogl daonismealgsr.oupThaet tphoesi7t2ivheocuornthraorlv,eCstP,grionudpucweedresisginginfiifciacnatntly increases in micronucleated means and standard errorsof 5P.C4Es4%in=bo0t.h37s%eaxensdas2c.o5m0p%a+re0d.3to3%thefovrethhieclmealcoenstraonlds, with ifnedmiavliedsu,alreaspneicmtailvedlayt.a aTrheefdoautnadsiunmTmaabrliezse2dtbhyroduogsheg7r.ouHipsatorreicparlesceonnttreodlidnaTtaabalree 1 and presented in Table 8. 150 CONCLUSION: nTmeahgreatttoievswtepmioanltteyhrcieharmlo,omuTas-t6ie3cm4ei2rc,yrtdohinrduoccnlyoettueissnaudsnusdcaeey.ratshiegnciofnidciatnitoinnsocfretahsiesiansmsiacyroannudcliseicoinnsbidoenreed CHV Study No.: 17073-0455 13 600342 160 REFERENCES: CORNING Hazleton aDcuonnntertotl,.C.JW..A:.m.AStmautlitsti.plAesscoomcp,a5r0i:s1o0n9s6-p1ro1c2e1d,u1r9e5f5o.r comparing several treatments with Dunnett, C.W.: 491, 1964. New tables for multiple comparisons witah control. Biometrics, 20:482- aHnedddSlael,aJm.oAn.,e,HiMt.eF,.M:, ThKieriknhdaurc,tiBo.n,oLfarmsiecnr,onKu.,clMeaicaGsreagmoera,suJ.rTe.o, fNegweenlolt,oxGi.ciWt.y. MutationRes., 123:61-118, 1983. Schmid, W.:. The micronucleus test. Mutation Res, 31:9-15, 1975. MSucthamgiedn,sW:.:PriTnhceipmliecsraonnducMleetuhsotdesstffoorrTchyetiorgeDneetteicctiaonna,lyVsoils.. Chemical 4 (A. Hollaender, ed). Plenum, pp. 31-53, 1976. YWoirnke,r,SBe.cJo.:ndStEadtiitsitoinc,al Principles 1971. in Experimental Design, McGraw-Hill, New CHV Study No.: 17073-0455 14 00343 `CORNING Hazleton 17.0 EXPERIMENT DATA TABLES CHV Study No.: 17073-0455 1s 00344 CORNINGHazleton SPONSOR: 3 Corporation TEST ARTICLE:T-6342 MICRONUCLEUSTDAABTLAE S1UMMARY TABLE ASSAY:17073 TREATMENT cowaoLs vEIGE TOSTIEGE DOSE HATRIVNEEST (Rr) acer Wh 80.0 mk he MEAN O*%FMI1C0R0O0NUPCELREAATNEIDMALPC%EsS.2. aes FEMALES TOTAL RAMTEIAONPCE5:.NEC.E MALES FEMALES oaisom 542037 0-0220.02 1302003 oonto.oz | 0s1to.0s amiose | cette 0.520. oe sens TT ARTICLE 1250 make he "hr 7h BO ml he "wh he 000 make he "wn nr 0.284 0.05 0.000.00 oossom 0.022004 cmon omen 0.0620.06 custo ose 0.002000 0.0220.02 e-0120.02 0.0020.02 .0220.02 o0620.00 0.0020.04 0.062002 0.032000 oa420.05 | 049x000 0.10.01 | 0.68 to.0n ooe20.0: | 0360.08 0.0020.02 | 0.6920.07 0.0220.01 | 0.7920.00 omzo0 | ourzo.0r 0.0020.03 | 0.00%0.08 0.1020.00 | o36%0a0 0.0920.03 | 0720.04 07s sour 0.74 0.08 0.3920.08 0.602008 ous 20.01 o.6to.0 0.75 0.00 0.63% 0.08 0.2620.050 "Significantly different from the corresponding vehicle sentrel. pO 0% CHV Study No.: 17073-0455 16 00345 `CORNINGHazleton MICRONUGLEUS TEST T-ABILNEDI2VIDUAL ANIMAL DATA SPONSOR3:M Corporation TEST ARTICLE:T-6342 HEASSAY No.:17073 ANDHAL vaad TIO _ SREASHENT TnUumer(lPoSoEpe) FOEpcNpNinCcEe _-- VERICLE CONTROL acer. wwee 3 00.3342 EwmHaw 21 ooslea ost POSITIVE CONTROL CP 80.0 mks 9 ae u61s 00.5709 m ms asz nw oeste os Test rier 0 aks ww wre d34 0o0.7s6s87 m ma 33 boeigs m0 wk wwes 21 o[l Hmnei o2 0B0e.7920 FR. we oo 0.51 _-- Fm wSs o1 7pasee NoPCMEN= PPCoMENlsyc==hrMNoiimccarrtooinncuucclelereuyasttherdocFyEteS NCE=Normochromatic erythrocyte CHV Study No.: 17073-0455 00346 1" `CORNINGHazleton nrcRowcLeus Testa"nTepiv3iouaL ANIMAL baa SPONSOR3:M Corporation TEST ARTICLE: T-6342 CATssayewwo.i170rmer73 momoemn PCOBE s pmmCo --__--o--m csr rs (000) PeE:NeE I -------- ma oe s oor oooonnnne osm coma woe mis mos me ow om Ben ol mans we wm FFaErso ae Bo wm moo mwmoe0 aas m FFHH odu wx Fo wHe s0 oenm e _-- e m ae oaal NPWGEoE N=oPrPmC0ooSlcyhc=+ehoWiWoimincseertrtoioimcmeuceeilareesynnyseeshehrdooccByyetoee CHVStudy No.: 17073-0-455 00347 18 : `CORNINGHazleton SPONSOR3M:MICRCOoNrUpCoLrEaUtSionTEST T-ABILNEDI4VIDUAL ANIMAL bATA TEST ARTICLE:T-6342 ASSAY No.:17073 TREATIES hAomza TPOCEE GaEAnTsIC oo oun waver ace Test aamzeus _-- we wa soo akg 000 mung s nm0oo oo0 ooondut FmEao on44 mwwees o oo on n0.51 Ea E o In H EwFHrr oo0le. omei 5 oh NPoCMEN= CP"EoMASlYnyic=m=harliMoeeimccafrotooniuncunudccelirdeoyeastathderdoc0ytse NCE-Normocheomatic erytheacyie CHV Study No.: 17073-0-455 00348 19 `CORNINGHazleton wicRowcLzvs Test maHabv5inuL aviv oan SPONSOR: Corporation Test AnTroLE T6242 T ASSAYEA0.Tr 1E1N7073 eme Mek r foze e TIO _ J-P_-- ------ (ooo)"NE -- 202 = oWYy= HnicraonaciTEeotnhRsroc3 yte NE om GeeR Cae CHV Study No.:17073-0455 00349 20 `CORNING Hazleton WICROWUCLEuS TEST asReBIVIOUAL ANIMAL DATA SPONSOR3:H Corporation Test AntroLET6302 ASSAY wo.117073 --_-- EATEN MowmgTsAR PoLze y(rATaIC e on wa mas o (logy) PCE:NCE ee "Animalce rfouond ndseeane d NPRCoeEEhm=noFproomlReycahhenR mmaerciies sayrY oaheraoccryctse CHV Study No.: 17073-0455 00350 21 `CORNINGHazleton wicRowcizus Testm"anTHeDIVIDUAL ANDHAL DATA SPONSOR3:M Corporation TEST ARTICLE T6342 TACSSAmTYReEwoAm.T:Ie1E7Se073 mNommex PCOEBs SmTmE _ I _-- ---- 0(100000)0POE:NCE mEATEE 0 wm emmeoofs0 oeae E eoEs om we wk Fmmreos1 oenw m moososoa 0 wa Ro mmS s0 ea e _-- eE Wn O E ew NETCH+ Pe"EAlSnyicn=haNilicosenviffotoniumutned]agndaeyecsaedhersocVyetee RCENormachepaatie aryhencr CHV Study No.: 17073-0-455 00351 22 . `CORNINGHazleton TABLE 8 MOUSE MICRONUCLEUS HISTORICAL CONTROL DATA 2/95 THROUGH 9/95 % MWEIACNRONOFUCL1E00A0TEPDERPCAEN:IMpAerL 1000 PGE * S.2. RATIO FCETNCE MEAN 5.2. TooLEd vanzoLr cowrRaL MALES FEMALES TOTAL MALES FEMALES Ed ax AVG 0.00 0.26 0.08 0.05 0.00 0.16 0.06%0.04 0.01 0.32 0.18 0.0720.04 | 0.82 0.56 0.43 0.3 1.08 0.61% 0.14 " " " "0 " CryocslzoTpahvoespchonaTnRiodre.. 0 mg/kg. a 12 x 5.46 1.30 6.36 10 3.8 0.44 0.72 0.4 0.01 AV n 3.252094 2 3.002105 2 3320.81 | 0.58 0.00 a a 0.62 20.1 2 CHV Study No.: 17073-0-455 00352 23